Compile Data Set for Download or QSAR
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Found 7 of ki data for polymerid = 50003294
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50314845(3'-(4-Chlorophenyl-1,2,3-triazol-1-yl)-3'-deoxy-be...)
Affinity DataKi:  12nMAssay Description:Competitive inhibition of human recombinant mitochondrial thymidine kinase 2 using ATP as substrate by Lineweaver-Burk plottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50314848(3'-hexanoylamino-3'-deoxythymidine | CHEMBL1089836)
Affinity DataKi:  150nMAssay Description:Inhibition of thymidine kinase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50200995(1-[6-[1,1-(diphenyl)-1-(4-pyridyl)methoxy]hexyl]th...)
Affinity DataKi:  290nMAssay Description:Inhibition of TK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50314845(3'-(4-Chlorophenyl-1,2,3-triazol-1-yl)-3'-deoxy-be...)
Affinity DataKi:  410nMAssay Description:Uncompetitive inhibition of human recombinant mitochondrial thymidine kinase 2 using thymidine as substrate by Lineweaver-Burk plottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118490(1-[(Z)-4-(triphenylmethoxy)-2-butenyl]thymine | 5-...)
Affinity DataKi:  500nMAssay Description:Inhibition of TK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50206491(1-beta-D-arabinofuranosyl-5-(2-bromovinyl)uracil |...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of thymidine kinase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase 2, mitochondrial(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50375778(CHEMBL221982)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed